研究者データベース - 白井　隆一

シライ　リュウイチ SHIRAI Ryuichi
白井　隆一

所属同志社女子大学薬学部医療薬学科

職種特別任用教授

著書・論文歴
著書	有機化学explorer (共著) 2009/08
著書	ベーシック薬学教科書シリーズ５　有機化学,128-173頁 (共著) 2008/12
著書	ブラウン・プーン基本有機化学 (共著) 2006/05/10
論文	Synthesis of Novel Pseudo-Enantiomeric Phase-Transfer Catalysts from Cinchona Alkaloids and Application to the Hydrolytic Dynamic Kinetic Resolution of Racemic 3-Phenyl-2-oxetanone（査読付） Chem. Pharm. Bull. 72 (10),913-916頁 (共著) 2024/10
論文	Hydrolytic dynamic kinetic resolution of racemic 3-phenyl-2-oxetanone to chiral tropic acid（査読付） RSC Advances 14,6121-6126頁 (共著) 2024/02
論文	Enantioselective [2,3]-Wittig rearrangement of carboxylic acid derived enolates by tetradentate chiral lithium amide（査読付） Synlett Vol. 2023 (No. 34),1727-1731頁 (共著) 2023/03
論文	官能基化されたNHC配位子の開発と触媒的アリール化反応へ適用有機合成化学協会誌 Vol.73 (No.4),p.361-371頁 (共著) 2015/04
論文	Efficient synthesis of 3-arylphthalides using palladium-catalyzed arylation of aldehydes with organoboronic acids（査読付） The Journal of Organic Chemistry Vol.74 (No.23),9210-9213頁 (共著) 2009/10
論文	Palladium-catalyzed 1,2-addition of potassium aryl- and alkenyltrifluoroborates to aldehydes using thioether-imidazolium carbine ligands（査読付） The Journal of Organic Chemistry Vol.73 (No.17),6939-6942頁 (共著) 2008/08
論文	Design and synthesis of N-alkyl-oxindolydene acetic acids as a new class of potent Cdc25A inhibitors（査読付） Bioorganic and Medicinal Chemistry Letters Vol.18 (No.11),3350-3353頁 (共著) 2008/06
論文	A novel route for the construction of Taxol ABC-ring framework: skeletal rearrangement approach to AB-ring and intramolecular aldol approach to C-ring（査読付） Tetrahedron Vol.64 (No.18),4051-4059頁 (共著) 2008/04
論文	Direct asymmetric aldol reactions catalyzed by L-proline-2,4,6-trinitroanilide（査読付） Tetrahedron Letters Vol.49 (No.15),2402-2406頁 (共著) 2008/04
論文	An acid-catalyzed ring-switch reaction of lactams to lactones:concise synthesis of 2,4-dialkyl-3-hydroxybutanolides（査読付） Tetrahedron Vol.64 (No.14),3133-3140頁 (共著) 2008/03
論文	Efficient 1,2-addition of aryl- and alkenylboronic acids to aldehydes catalyzed by the palladium/thioether-imidazolium chloride system（査読付） The Journal of Organic Chemistry Vol.73 (No.4),1597-1600頁 (共著) 2008/01
論文	Design and Synthesis of Thioether-Imidazolium Chlorides as Efficient Ligands for Palladium-Catalyzed Suzuki-Miyaura Coupling of Aryl Bromides with Arylboronic Acids（査読付） Tetrahedron Vol.63 (No.38),9393-9400頁 (共著) 2007/09
論文	Design and Synthesis of Novel C₂-Symmetric Chiral Piperazines and an Application to Asymmteric Acylation of-Symmteric 1,2-diols（査読付） Organic Letters Vol.8 (No.2),6139-6142頁 (共著) 2006/12
論文	Design and synthesis of novel Cdc25A inhibitors having phosphate group as a hydrophilic residue（査読付） Bioorganic and Medicinal Chemistry Letters Vol.14,4339-4342頁 (共著) 2004/08
論文	Design and synthesis of dysidiolide analogs from vitamin D3: novel class of Cdc25A inhibitors（査読付） Bioorganic and Medicinal Chemistry Letters Vol.14,3291-3294頁 (共著) 2004/06
論文	Diastereoselective synthesis of D- and L-myo-inositol 3,4,5,6-tetrakis-phosphates from D-glucose via dihydroxylation of (+)-conduritol B derivatives（査読付） Chemical and Pharmaceutical Bulletin Vol.52,727-732頁 (共著) 2004/06
論文	Synthesis of L-α-phosphatidyl-D-myo-inositol 3,5-bisphosphate from D-glucose（査読付） Tetrahedron Letters Vol.42,9195-9198頁 (共著) 2001/11
論文	リチウムエノラートの触媒的不斉反応マテリアル　インテグレーション Vol.14,68-71頁 (共著) 2001/05
論文	Synthesis of the novel analogs of dysidiolide and their structure-activity relationship（査読付） Bioorganic and Medicinal Chemistry Letters Vol.10,2571-2574頁 (共著) 2000/10
論文	微小管機能を制御する天然有機化合物：コルヒチン部位に結合するコンブレタスタチン及びキュラシンA関連化合物の合成と構造活性相関薬学雑誌 Vol.120,875-889頁 (共著) 2000/10
論文	Separation of phosphatidylinositol 4-phosphate from a mixture with phosphatidylserine and phosphatidylinositol by Sep-Pak C18 cartridge（査読付） Biological and Pharmaceutical Bulletin Vol.23,1088-1089頁 (共著) 2000/09
論文	Evidence that 3’-phosphorylated polyphosphoinositides are generated at the nuclear surface: use of immunostaining techniqe with monoclonal antibodies specific for PI 3,4-P2（査読付） FEBS Letters Vol.473,222-226頁 (共著) 2000/04
論文	Phosphorylation of unnatural phosphatidylinositols with phosphatidylinositol 3-kinase（査読付） Tetrahedron Vol.56,2603-2614頁 (共著) 2000/04
論文	Quantification of phosphatidylinositol 3,4,5-trisphosphate by liposome lysis assay with specific monoclonal antibodies（査読付） Analytical Biochemistry Vol.285,270-273頁 (共著) 2000/04
論文	Concise asymmetric synthesis of dysidiolide（査読付） Tetrahedron Letters Vol.41,2111-2114頁 (共著) 2000/02
論文	Synthesis of a novel class of cdc25A inhibitor from Vitamin D3（査読付） Bioorganic and Medicinal Chemistry Letters Vol.10,615-617頁 (共著) 2000/02
論文	The structural requirement of phosphatidyl-inositols as substrate of phosphatidylinositol 3-kinase（査読付） Tetrahedron Letters Vol.40,1693-1696頁 (共著) 1999/12
論文	らん藻Lingbya majusculaから単離された有糸分裂阻害剤Curacin Aの合成有機合成化学協会誌 Vol.57,58-66頁 (単著) 1999/06
論文	Novel small molecule nonpeptide aminopeptidase N inhibitors with a cyclic imide skeleton Journal of Enzyme Inhibition Vol.14,265-271頁 (共著) 1999/01
論文	Synthesis of the diacylglycerol analogs of phosphatidylinositol 3,4,5-trisphosphate（査読付） Tetrahedron Letters Vol.39,9485-9488頁 (共著) 1998/11
論文	Synthesis of 6-amylsalicylic acid from 3-anisaldehyde: conversion of phthalide to thiophtalide by aluminum halide-butanethiol（査読付） Tetrahedron Letters Vol.39,7307-7308頁 (共著) 1998/09
論文	Antimitotic combretadioxolane with potent antitumor activity against multi-drug resistant cells（査読付） Bioorganic and Medicinal Chemistry Letters Vol.8,1997-2000頁 (共著) 1998/07
論文	Tumor necrosis facter-alpha production enhancing activity of substituted 3’-methylthalidomide: influence of substitutents at the phthaloyl moiety on the activity and stereoselectivity（査読付） Chemical and Pharmaceutical Bulletin Vol.46,1165-1168頁 (共著) 1998/07
論文	Collisionally activated dissociation of 13-membered peptides, ustiloxins and phomopsins（査読付） Journal of Mass Spectrometry Society of Japan Vol.46,495-501頁 (共著) 1998/06
論文	Isolation and structure of an antimitotic cyclic peptide, ustiloxin F: chemical interrelation with a homologous peptide, ustiloxin B（査読付） Journal of Antibiotics Vol.51,418-422頁 (共著) 1998/04
論文	Synthesis and anti-tubulin activity of ustiloxin D derivatives（査読付） Journal of Antibiotics Vol.51,423-427頁 (共著) 1998/04
論文	Sequence selective interaction between nucleotides and intercalators bound to water soluble dextran: an application to the affinity chromatography of dinucleotides（査読付） Nucleosides and Nucleotides Vol.17,593-601頁 (共著) 1998/03
論文	Specific detection of phosphatidylinositol 3,4,5-trisphosphate binding proteins by the PIP3 analogue beads: an application for rapid purification of the PIP3 binding proteins（査読付） Biochimica et Biophysica Acta Vol.1402,292-302頁 (共著) 1998/03
論文	Synthetic study of novel ustiloxin analogs: benzylic oxidation of 13-membered cyclic peptide by lead tetraacetate（査読付） Heterocycles Vol.47,163-166頁 (共著) 1998/01
論文	Phosphorylation of the immunosuppressant FK506-binding protein FKBP52 by casein kinase II (CK2): regulation of HSP90-binding activity of FKBP52（査読付） Proceedings of the National Academy of Sciences, USA Vol.94,14500-14505頁 (共著) 1997/12
論文	Design and synthesis of the side chain analogs of curacin A（査読付） Bioorganic and Medicinal Chemistry Letters Vol.7,2657-2660頁 (共著) 1997/10
論文	Efficient asymmetric synthesis of phosphatidyl-D-myo-inositol 3,4,5-trisphosphate（査読付） Chemical and Pharmaceutical Bulletin Vol.45,1521-1523頁 (共著) 1997/09
論文	Stereoselective reactions. 25. Enantioselective deprotonation of prochiral 4-substituted cyclohexanones by chiral chelated lithium amides（査読付） Tetrahedron Vol.53,5963-5972頁 (共著) 1997/08
論文	A mild and selective deprotection of p-methoxybenzyl (PMB) ether by magnesium bromide diethyl etherate-methyl sulfide（査読付） Tetrahedron Letters Vol.38,1443-1446頁 (共著) 1997/02
論文	Synthesis of 5-[(2,5-dihydroxy- benzyl)amino]- salicylic acid analogs as potent EGF-R protein tyrosine kinase inhibitors（査読付） Bioorganic and Medicinal Chemistry Letters Vol.7,365-368頁 (共著) 1997/02
論文	A target of phosphatidylinositol 3,4,5-trisphosphate with a zinc finger motif similar to that of the ADP ribosylation factor GTPase activating protein and two pleckstrin homology domains（査読付） Europian Journal of Biochemistry Vol.245,513-516頁 (共著) 1997/01
論文	Non-intercalative and sequence selective interaction between four intercalative reagents and dinucleotides Nucleic Acids Symposium Series Vol.37,79-80頁 (共著) 1997/01
論文	Synthesis of conformationary restricted combretastatins（査読付） Heterocycles Vol.46,145-148頁 (共著) 1997/01
論文	Synthetic study on curacin A: a novel antimitotic agent from the cyanobacterium Lyngbya majuscula（査読付） Tetrahedron Vol.52,14543-14562頁 (共著) 1996/11
論文	Efficient asymmetric synthesis of cis-2-methylcyclopropanecarboxylic acid（査読付） Tetrahedron Vol.52,13327-13338頁 (共著) 1996/10
論文	Coordination of alkali metal cation to oxygen functions to form adduct ion in fast atom bombardment mass spectrometry（査読付） Tetrahedron Vol.52,9017-9024頁 (共著) 1996/07
論文	Asymmetric total synthesis of curacin A（査読付） Tetrahedron Letters Vol.37,4397-4400頁 (共著) 1996/06
論文	Facile asymmetric synthesis of the myo-inositol derivative from diethyl 2,3-O-isopropylidene-D- tartrate（査読付） Tetrahedron Letters Vol.37,886-887頁 (共著) 1996/02
論文	Tremorgenic indole alkaloids. 9. asymmetric construction of an Advanced F-G-H-ring lactone precursor for the synthesis of penitrem D（査読付） Journal of Organic Chemistry Vol.60,7837-7848頁 (共著) 1995/11
論文	Synthesis of 1-O-alkyl- and 1-O-acyl-myo-inositol 3,4,5-trisphosphates as novel analogues of phosphatidyl-myo-inositol 3,4,5-trisphosphate（査読付） Bioorganic and Medicinal Chemistry Letters Vol.5,2263-2266頁 (共著) 1995/10
論文	Synthetic study of curacin a: synthesis of partial structure of curacin A and elucidation of the absolute stereochemistry at the methylcyclopropylthiazoline moiety（査読付） Tetrahedron Letters Vol.36,5765-5768頁 (共著) 1995/08
論文	Cytotoxicity and DNA-binding property of non-diynene class of dynemicins and aza-anthraquinones（査読付） Nucleic Acids Symposium Series Vol.34,151-152頁 (共著) 1995/01
論文	Synthetic approach toward the minimal active structure of phomopsin-ustiloxin class of antibiotics: construction of 13-membered cyclic peptide skeleton（査読付） Heterocycles Vol.41,9-12頁 (共著) 1995/01
論文	DNA-binding ability of non-diynene class of dynemicins and aza-anthraquiqnones（査読付） Bioorganic and Medicinal Chemistry Letters Vol.4,2377-2382頁 (共著) 1994/10
論文	Stereoselective reactions. 22. Design and synthesis of chiral chelated lithium amides for enantioselective reactions（査読付） Chemical and Pharmaceutical Bulletin Vol.42,690-693頁 (共著) 1994/03
論文	Synthesis and anti-tubulin activity of aza-combretastatins（査読付） Bioorganic and Medicinal Chemistry Letters Vol.4,699-704頁 (共著) 1994/03
論文	Interaction of marine toxin dolastatin 10 with porcine brain tubulin: competitive inhibition of rhizoxin and phomopsin A binding（査読付） Chemico-Biological Interactions Vol.93,175-183頁 (共著) 1994/01
論文	Enantioselective deprotonation of the meso-forms of 2,6- and 3,5-dimethylcyclohexanones（査読付） Heterocycles Vol.30,307-310頁 (共著) 1990/01
論文	Enantioselective deprotonation of monoacetals of bicyclo[3,3,0]octane-3,7-dione. an approach to the asymmetric synthesis of chiral synthons for carbacyclins（査読付） Tetrahedron Letters Vol.30,7221-7224頁 (共著) 1989/12
論文	Improved syntheses of two 3-deoxyald-2-ulosonic acids (KDN, KDO) by condensation of oxalacetic acid with aldoses followed by Ni²⁺ catalyzed decarboxylation（査読付） Tetrahedron Letters Vol.30,2263-2264頁 (共著) 1989/03
論文	Thermal rearrangement of N-acetyl-N-nitrosoneuraminic acid derivative: synthesis of 3-deoxy-D- nonulosonic acid (KDN)（査読付） Tetrahedron Letters Vol.29,4449-4452頁 (共著) 1988/10
論文	キラルなリチウムアミドを用いる不斉脱プロトン化反応化学 (化学同人、京都) Vol.41,546-547頁 (共著) 1986/08
論文	キラル塩基を用いるエナンチオ選択的脱プロトン化反応の開発（査読付）博士学位論文 (単著) 1986/03
論文	Enantioselective deprotonation by chiral lithium amide bases: asymmetric synthesis of trimethylsilyl enol ethers from 4-alkylcyclohexanones（査読付） Journal of the American Chemical Society Vol.108,543-545頁 (共著) 1986/02
論文	Studies on tetra- hydroisoquinolines. XXV. A synthesis of 4-aryl-1,2,3,4-tetrahydroisoquinolines; total synthesis of (±)-cherylline（査読付） Chemical and Pharmaceutical Bulletin Vol.33,3107-3112頁 (共著) 1985/04
論文	Studies on tetrahydroisoquinolines. XXI. A synthesis of (±)-1-hydroxy-2-methoxy-homoproaporphine and stereochemistry of 4-oxygenated 1,2,3,4-tetrahydroisoquinolines（査読付） Chemical and Pharmaceutical Bulletin Vol.31,4236-4246頁 (共著) 1983/06
論文	A facile synthesis of 4-aryl-1,2,3,4-tetrahydroisoquinolines: A total synthesis of (±)-cherylline（査読付） Heterocycles,1945-1950頁 (共著) 1983/05
その他	薬学6年制でこそ充実した卒業研究を薬事日報 (単著) 2006/04/12